| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
SJ-GBM2 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
HB-1643 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
NB-EBc1 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
CHLA-90 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
CHLA-136 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
NALM-6 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
COG-LL-317 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
RS4;11 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
MOLt-4 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
CCRF-CEM GM |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
CCRF-CEM-SY |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
Kasumi-1 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
Karpas-299 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell viability |
DIMSCAN |
N/A nM |
Ramos-RA1 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell proliferation in tumor tissue |
Tumour volume |
60.00 mg/kg |
KT-6 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell proliferation in tumor tissue |
Tumour volume |
60.00 mg/kg |
KT-11 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell proliferation in tumor tissue |
Tumour volume |
60.00 mg/kg |
KT-10 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on cell proliferation in tumor tissue |
Tumour volume |
60.00 mg/kg |
KT-8 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
20.00 mg/kg |
KT-10 |
Homo sapiens |
|
STAT3 |
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
20.00 mg/kg |
KT-10 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
10.00 mg/kg |
KT-10 |
Homo sapiens |
|
STAT3 |
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
10.00 mg/kg |
KT-10 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
20.00 mg/kg |
KT-13 |
Homo sapiens |
|
STAT3 |
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
20.00 mg/kg |
KT-13 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
10.00 mg/kg |
KT-13 |
Homo sapiens |
|
STAT3 |
|
| AZD1480 |
Influence on protein level in tumor tissue |
Western Blot |
10.00 mg/kg |
KT-13 |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on cell viability |
MTT |
5.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on cell viability |
MTT |
10.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on cell viability |
MTT |
20.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
5.00 µM |
PANC-I |
Homo sapiens |
|
p-STAT3 (Y705) |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
10.00 µM |
PANC-I |
Homo sapiens |
|
p-STAT3 (Y705) |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
20.00 µM |
PANC-I |
Homo sapiens |
|
p-STAT3 (Y705) |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
30.00 µM |
PANC-I |
Homo sapiens |
|
p-STAT3 (Y705) |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
5.00 µM |
PANC-I |
Homo sapiens |
|
STAT3 |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
10.00 µM |
PANC-I |
Homo sapiens |
|
STAT3 |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
20.00 µM |
PANC-I |
Homo sapiens |
|
STAT3 |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
30.00 µM |
PANC-I |
Homo sapiens |
|
STAT3 |
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
5.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
10.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
20.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
30.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
5.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
10.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
20.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
30.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
5.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
10.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
20.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on protein levels |
Western Blot |
30.00 µM |
PANC-I |
Homo sapiens |
|
|
|
| Benzyl isothiocyanate |
Influence on STAT3 target expression |
RT-PCR |
10.00 µM |
PANC-I |
Homo sapiens |
|
|
|