Cyclometalated rhodium(III) complex 12 |
Influence on protein binding |
Cell-free assay |
30.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein binding in presence of EGF |
Fluorescence polarization assay |
0.30 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein binding in presence of EGF |
Fluorescence polarization assay |
1.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein binding in presence of EGF |
Fluorescence polarization assay |
3.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein binding in presence of EGF |
Fluorescence polarization assay |
10.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein binding in presence of EGF |
Fluorescence polarization assay |
30.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
3.00 µM |
A375 |
Homo sapiens |
|
p-STAT3 (Y705) |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
10.00 µM |
A375 |
Homo sapiens |
|
p-STAT3 (Y705) |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
20.00 µM |
A375 |
Homo sapiens |
|
p-STAT3 (Y705) |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
3.00 µM |
A375 |
Homo sapiens |
|
STAT3 |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
10.00 µM |
A375 |
Homo sapiens |
|
STAT3 |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
20.00 µM |
A375 |
Homo sapiens |
|
STAT3 |
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
3.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
10.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Western Blot |
20.00 µM |
A375 |
Homo sapiens |
|
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Immunohistochemistry |
75.00 mg/kg |
A375(xenograft) |
Mus musculus |
BALB/c |
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Immunohistochemistry |
75.00 mg/kg |
A375(xenograft) |
Mus musculus |
BALB/c |
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on protein activity |
Immunohistochemistry |
75.00 mg/kg |
A375(xenograft) |
Mus musculus |
BALB/c |
|
|
Cyclometalated rhodium(III) complex 12 |
Influence on blood flow |
Laser Doppler flowmetry |
75.00 mg/kg |
A375(xenograft) |
Mus musculus |
BALB/c |
|
|
Dasatinib |
Influence on gene expression |
qRT-PCR |
3.30 nM |
K562 |
Homo sapiens |
|
STAT5A |
|
Dasatinib |
Influence on gene expression |
qRT-PCR |
3.30 nM |
K562 |
Homo sapiens |
|
STAT5B |
|
Dasatinib |
Influence on protein activity |
Western Blot |
3.30 nM |
K562 |
Homo sapiens |
|
STAT5A |
|
Dasatinib |
Influence on protein activity |
Western Blot |
3.30 nM |
K562 |
Homo sapiens |
|
STAT5B |
|
Dasatinib |
Influence on protein activity |
Western Blot |
3.30 nM |
K562 |
Homo sapiens |
|
|
|
Dasatinib |
Influence on cell viability |
Colony formation assay |
10.00 nM |
MPN |
Homo sapiens |
|
|
|
Dasatinib |
Influence on cell viability |
Colony formation assay |
1.00 nM |
ET |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
p-STAT5 |
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
p-STAT5 |
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
p-STAT5 |
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
STAT5 |
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
STAT5 |
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
STAT5 |
|
Dasatinib |
Influence on protein activity |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity |
Western Blot |
100.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|
Dasatinib |
Influence on protein activity in presence of Ruxololitinib |
Western Blot |
10.00 nM |
BaF3 JAK2 V617F |
Homo sapiens |
|
|
|