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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 0.50 µM MO4 Mus musculus
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 1.00 µM MO4 Mus musculus
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 5.00 µM MO4 Mus musculus
AZD1480 Function of myeloid-derived suppressor cells 30.00 mg/kg MO4 (xenograft) Mus musculus c57BL/6
AZD1480 Influence on cell proliferation Flow cytometry 1.75 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 1.50 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 1.25 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 1.00 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.75 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.50 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.25 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.10 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.05 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.03 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation Flow cytometry 0.01 µM Splenocytes Mus musculus
AZD1480 Influence on cell proliferation ELISA 1.50 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 1.25 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 1.00 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 0.75 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 0.50 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 0.25 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 0.10 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on cell proliferation ELISA 0.05 µM CD 8+ T cells Homo sapiens
AZD1480 Influence on protein activity Western Blot 0.10 µM HD-LM2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM HD-LM2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM HD-LM2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM HD-LM2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM HD-LM2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM HD-LM2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM HD-LM2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM HD-LM2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM L-428 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM L-428 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM L-428 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM L-428 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM L-428 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM L-428 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM L-428 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM L-428 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM KM-H2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM KM-H2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM KM-H2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM KM-H2 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM KM-H2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM KM-H2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM KM-H2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 5.00 µM KM-H2 Homo sapiens STAT1
AZD1480 Influence on protein activity Western Blot 0.10 µM L-540 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 0.50 µM L-540 Homo sapiens p-STAT1
AZD1480 Influence on protein activity Western Blot 1.00 µM L-540 Homo sapiens p-STAT1