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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
AZD1480 Influence on protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice p-STAT3 (Y705)
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice p-STAT3 (Y705)
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice p-STAT3 (Y705)
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice p-STAT3 (Y705)
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice STAT3
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice STAT3
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice STAT3
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice STAT3
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on late protein activity in tumor tissue Western Blot 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on tumor growth Histological staining 30.00 mg/kg KCNR (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on tumor growth Histological staining 30.00 mg/kg SY5Y (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on tumor growth Histological staining 30.00 mg/kg Rh18 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on tumor growth Histological staining 30.00 mg/kg TC32 (xenograft) Mus musculus athymic nude mice
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 0.50 µM MO4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 0.50 µM K1735-C4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 0.50 µM 1087-mel Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 1.00 µM MO4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 1.00 µM K1735-C4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 1.00 µM 1087-mel Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 5.00 µM MO4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 5.00 µM K1735-C4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 5.00 µM 1087-mel Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 10.00 µM MO4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 10.00 µM K1735-C4 Mus musculus
AZD1480 Influence on apoptosis Flow cytometry- annexin V staining 10.00 µM 1087-mel Mus musculus
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 0.50 µM MO4 Mus musculus p-STAT3
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 1.00 µM MO4 Mus musculus p-STAT3
AZD1480 Influence on protein activity in presence of IL-6 Western Blot 5.00 µM MO4 Mus musculus p-STAT3