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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (JAK2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (JAK2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (JAK2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (JAK3-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (JAK3-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (Tyk2-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (Tyk2-JH1) Homo sapiens STAT3
Brevilin A Influence on tumor growth Tumor volume and weight, mouse body weight 4.50 mg/kg A375 Mus musculus
Brevilin A Influence on tumor growth Tumor volume and weight, mouse body weight 9.00 mg/kg A375 Mus musculus
Brevilin A Influence on protein levels in tumor tissue Western Blot 4.50 mg/kg A375 Mus musculus pTyr705-STAT3
Brevilin A Influence on protein levels in tumor tissue Western Blot 9.00 mg/kg A375 Mus musculus pTyr705-STAT3
Brevilin A Influence on protein levels in tumor tissue Western Blot 4.50 mg/kg A375 Mus musculus STAT3
Brevilin A Influence on protein levels in tumor tissue Western Blot 9.00 mg/kg A375 Mus musculus STAT3
Brevilin A Influence on cell viability MTT 0.50 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 1.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 2.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 4.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 8.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 12.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 16.00 µM A375 Homo sapiens
Brevilin A Influence on cell viability MTT 0.50 µM A2058 Homo sapiens
Brevilin A Influence on cell viability MTT 1.00 µM A2058 Homo sapiens
Brevilin A Influence on cell viability MTT 2.00 µM A2058 Homo sapiens
Brevilin A Influence on cell viability MTT 4.00 µM A2058 Homo sapiens
Brevilin A Influence on cell viability MTT 8.00 µM A2058 Homo sapiens
Brevilin A Influence on cell viability MTT 12.00 µM A2058 Homo sapiens