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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Piperlongumine Influence on protein activity Western Blot 2.50 µM 786-O Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 5.00 µM 786-O Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 10.00 µM 786-O Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 10.00 µM MKN45 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 20.00 µM MKN45 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 40.00 µM MKN45 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 1.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 3.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 10.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 30.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 100.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein phosphorylation Flow cytometry 300.00 µM Kasumi 1 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 0.10 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 0.30 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 1.00 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 3.00 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 10.00 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 30.00 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 100.00 µM MDA-MB-468 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 0.10 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 0.30 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 1.00 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 3.00 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 10.00 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 30.00 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity (with and without ligand) Luminex assay 100.00 µM MDA-MB-231 Homo sapiens p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4400 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4849 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3613B Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3824 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4888 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4175 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3963 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft IBC3 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3807 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3204 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 2277 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4664 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3887 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3107 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 2665 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4169 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3561 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 4698 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3143 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3104 Mus musculus SCID/Beige nude mice p-STAT3
Piperlongumine Influence on cell apoptosis Luminex assay 30.00 µM patient derived xenograft 3611 Mus musculus SCID/Beige nude mice p-STAT3