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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Cryptotanshinone Influence on protein activity Western Blot 30.00 µM BxPC‑3 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 40.00 µM BxPC‑3 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM HCT116 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM HCT116 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 25.00 µM HCT116 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 50.00 µM HCT116 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM SW480 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM SW480 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 25.00 µM SW480 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 50.00 µM SW480 Homo sapiens STAT3
Cryptotanshinone Influence on protein activity Western Blot 1.25 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity Western Blot 2.50 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity Western Blot 20.00 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity in presence of pervanadate Western Blot 10.00 µM U251 Homo sapiens p-STAT3 (Y705)
Cryptotanshinone Influence on protein activity Western Blot 1.25 µM U251 Homo sapiens p-STAT3 (S727)
Cryptotanshinone Influence on protein activity Western Blot 2.50 µM U251 Homo sapiens p-STAT3 (S727)
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM U251 Homo sapiens p-STAT3 (S727)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM U251 Homo sapiens p-STAT3 (S727)
Cryptotanshinone Influence on protein activity Western Blot 20.00 µM U251 Homo sapiens p-STAT3 (S727)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM U251 Homo sapiens STAT3 (whole cell)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM U251 Homo sapiens STAT3 (nuclear)
Cryptotanshinone Influence on protein activity in transfected cells Western Blot 10.00 µM U251 SHP-2 Homo sapiens p-STAT3(Y705)
Cryptotanshinone Influence on protein activity in transfected cells Western Blot 5.00 µM U251 SHP-2 Homo sapiens p-STAT3(Y705)
Cryptotanshinone Influence on protein activity in transfected cells Western Blot 10.00 µM U251 TC-PTP Homo sapiens p-STAT3(Y705)
Cryptotanshinone Influence on protein activity in transfected cells Western Blot 10.00 µM U251 SHP-1 Homo sapiens p-STAT3(Y705)
Cryptotanshinone Influence on protein activity in tumor tissue Immunohistochemistry 30.00 mg/kg U87 (xenograft) Mus musculus BALB/c p-STAT3(Y705)
Cryptotanshinone Influence on protein activity in tumor tissue Immunohistochemistry 60.00 mg/kg U87 (xenograft) Mus musculus BALB/c p-STAT3(Y705)
Cryptotanshinone Influence on protein activity Western Blot 15.00 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 15.00 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 15.00 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 2.50 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 7.50 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 20.00 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 2.50 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 7.50 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 20.00 µM MKN45 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 2.50 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 5.00 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 7.50 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 10.00 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 20.00 µM HGC27 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 0.25 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 0.50 µM SGC7901 Homo sapiens p-STAT3 (Ser727)
Cryptotanshinone Influence on protein activity Western Blot 1.00 µM SGC7901 Homo sapiens p-STAT3 (Ser727)