Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
20.00 µM |
HEK293T (JAK3-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
5.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
7.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
10.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
12.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
15.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
17.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
20.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
pTyr705-STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
5.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
7.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
10.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
12.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
15.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
17.50 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
20.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on cell viability |
MTT |
0.50 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
1.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
2.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
4.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
8.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
12.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
16.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
0.50 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
1.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
2.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
4.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
8.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
12.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
16.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
0.50 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
1.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
2.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
4.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
8.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
12.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
MTT |
16.00 µM |
HaCaT |
Homo sapiens |
|
|
|
Brevilin A |
Influence on cell viability |
Annexin-V-PI dual staining |
1.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Annexin-V-PI dual staining |
2.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Annexin-V-PI dual staining |
3.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Annexin-V-PI dual staining |
1.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Annexin-V-PI dual staining |
2.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Annexin-V-PI dual staining |
3.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
1.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
2.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
3.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
1.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
2.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
3.00 µM |
A2058 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
1.00 µM |
A375 |
Homo sapiens |
|
|
|
Brevilin A |
Influence on apoptosis |
Western Blot |
2.00 µM |
A375 |
Homo sapiens |
|
|
|