Pacritinib |
Influence on protein activity |
Western Blot |
0.20 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
0.50 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
1.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
2.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
3.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
5.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
10.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
0.20 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
0.50 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
1.00 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
2.00 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
3.00 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
5.00 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
10.00 µM |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
0.20 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
0.50 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
1.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
2.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
3.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
5.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on protein activity |
Western Blot |
10.00 µM |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on survival |
Average survival |
100.00 mg/kg |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on survival |
Average survival |
100.00 mg/kg |
BT53 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on survival in tresence of TMZ |
Average survival |
100.00 mg/kg |
BT147 |
Homo sapiens |
|
|
|
Pacritinib |
Influence on survival in tresence of TMZ |
Average survival |
100.00 mg/kg |
BT53 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
10.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
25.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
50.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
75.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
100.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
10.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
25.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
50.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
75.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
MTS |
100.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
CellTiter-Glo luminescent assay |
100.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell viability |
CellTiter-Glo luminescent assay |
100.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell proliferation |
Flow cytometry |
30.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell proliferation |
Flow cytometry |
30.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell apoptosis |
Flow cytometry- annexin V binding and propidium iodide staining |
50.00 µM |
Jurkat |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on cell apoptosis |
Flow cytometry- annexin V binding and propidium iodide staining |
50.00 µM |
K562 |
Homo sapiens |
|
|
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
10.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
15.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
30.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
10.00 µM |
Jurkat |
Homo sapiens |
|
STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
15.00 µM |
Jurkat |
Homo sapiens |
|
STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
30.00 µM |
Jurkat |
Homo sapiens |
|
STAT1 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
10.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT3 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
15.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT3 |
|
Phloridzin docosahexaenoate |
Influence on protein activity in presence of IFNα |
Western Blot |
30.00 µM |
Jurkat |
Homo sapiens |
|
p-STAT3 |
|