| Dasatinib |
Influence on protein activity |
Western Blot |
0.01 µM |
HLF |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.10 µM |
HLF |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
1.00 µM |
HLF |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
10.00 µM |
HLF |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.00 µM |
Hep3B |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.01 µM |
Hep3B |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.10 µM |
Hep3B |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
1.00 µM |
Hep3B |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
10.00 µM |
Hep3B |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.00 µM |
HepG2 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.01 µM |
HepG2 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.10 µM |
HepG2 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
1.00 µM |
HepG2 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
10.00 µM |
HepG2 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.00 µM |
HT-17 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.01 µM |
HT-17 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.10 µM |
HT-17 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
1.00 µM |
HT-17 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
10.00 µM |
HT-17 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.00 µM |
Huh-7 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.01 µM |
Huh-7 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
0.10 µM |
Huh-7 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
1.00 µM |
Huh-7 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on protein activity |
Western Blot |
10.00 µM |
Huh-7 |
Homo sapiens |
|
|
|
| Dasatinib |
Influence on cell motility |
Invasion assay |
1.00 µM |
Sk-Hep1 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
0.10 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
1.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
10.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
30.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
100.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
0.10 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
1.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
10.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
30.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
100.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
0.10 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
1.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
10.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
30.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
100.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
0.10 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
1.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
10.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
30.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| ISS-610 prodrugs |
Influence on protein activity |
Western Blot |
100.00 µM |
MDA-MB-468 |
Homo sapiens |
|
|
|
| inS3-54A18 |
Influence on cell motility |
Colony formation assay |
20.00 µM |
CFU-GEMM |
Homo sapiens |
|
|
|
| inS3-54A18 |
Influence on cell motility |
Colony formation assay |
20.00 µM |
CFU-GM |
Homo sapiens |
|
|
|
| inS3-54A18 |
Influence on cell motility |
Colony formation assay |
20.00 µM |
BFU-E |
Homo sapiens |
|
|
|
| inS3-54A18 |
Influence on protein binding to DNA |
EMSA |
5.00 µM |
H1299 |
Homo sapiens |
|
STAT1 |
|
| inS3-54A18 |
Influence on protein binding to DNA |
EMSA |
13.00 µM |
H1299 |
Homo sapiens |
|
STAT1 |
|
