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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Toosendanin Influence on protein activity Luciferase reporter assay 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Luciferase reporter assay 50.00 nM HOS Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens p-STAT3(Y705)
Toosendanin Influence on protein activity Western Blot 50.00 nM HOS Homo sapiens p-STAT3(Y705)
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens p-STAT3(Y705)
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens p-STAT3(S727)
Toosendanin Influence on protein activity Western Blot 50.00 nM HOS Homo sapiens p-STAT3(S727)
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens p-STAT3(S727)
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens STAT3
Toosendanin Influence on protein activity Western Blot 50.00 nM HOS Homo sapiens STAT3
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens STAT3
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM HOS Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens STAT3(nucleus)
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens STAT3(cytoplasm)
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein translocation in presence of IL-6 Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein-DNA interaction EMSA 50.00 nM 143B Homo sapiens STAT3
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on expression of STAT3 target genes RT-PCR 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM 143B Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein activity Western Blot 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on protein-DNA interaction Chromatin immunoprecipitation assay 50.00 nM 143B Homo sapiens STAT3:Bcl2
Toosendanin Influence on protein-DNA interaction Chromatin immunoprecipitation assay 50.00 nM 143B Homo sapiens STAT3:VEGF
Toosendanin Influence on protein-DNA interaction Chromatin immunoprecipitation assay 50.00 nM 143B Homo sapiens STAT3:SOCS3
Toosendanin Influence on cell viability MTS Assay 50.00 nM 143B Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM HOS Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM MG63.2 Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM MG63 Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM DUNN Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM LM8 Homo sapiens
Toosendanin Influence on cell viability MTS Assay 50.00 nM hFOB1.19 Homo sapiens