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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens p-STAT3
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens STAT3
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens STAT3
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens STAT3
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 2.50 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 5.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on gene expression RT-qPCR 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity in presence of bortezomib Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on protein activity in presence of bortezomib Western Blot 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on ROS generation Flow cytometry 10.00 µM PNX0010 Homo sapiens
Piperlongumine Influence on cell viability Cell Titer Blue assay N/A µM PNX0010 Homo sapiens
Piperlongumine Influence on tumor growth Tumor volume 20.00 mg/kg PNX0010 (xenograft) Mus musculus C.B-17/Icr mice
Piperlongumine Influence on tumor growth Immunohistochemistry 20.00 mg/kg PNX0010 (xenograft) Mus musculus C.B-17/Icr mice