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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Dasatinib Influence on protein activity Western Blot 10.00 nM BaF3 JAK2 V617F Homo sapiens p-STAT5
Dasatinib Influence on protein activity Western Blot 100.00 nM BaF3 JAK2 V617F Homo sapiens p-STAT5
Dasatinib Influence on protein activity in presence of Ruxololitinib Western Blot 10.00 nM BaF3 JAK2 V617F Homo sapiens p-STAT5
Dasatinib Influence on protein activity Western Blot 10.00 nM BaF3 JAK2 V617F Homo sapiens STAT5
Dasatinib Influence on protein activity Western Blot 100.00 nM BaF3 JAK2 V617F Homo sapiens STAT5
Dasatinib Influence on protein activity in presence of Ruxololitinib Western Blot 10.00 nM BaF3 JAK2 V617F Homo sapiens STAT5
Dasatinib Influence on gene expression qRT-PCR 3.30 nM K562 Homo sapiens STAT5A
Dasatinib Influence on protein activity Western Blot 3.30 nM K562 Homo sapiens STAT5A
Dasatinib Influence on gene expression qRT-PCR 3.30 nM K562 Homo sapiens STAT5B
Dasatinib Influence on protein activity Western Blot 3.30 nM K562 Homo sapiens STAT5B