Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
1.25 µM |
CNE-2 |
Homo sapiens |
|
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
2.50 µM |
CNE-2 |
Homo sapiens |
|
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
5.00 µM |
CNE-2 |
Homo sapiens |
|
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
10.00 µM |
CNE-2 |
Homo sapiens |
|
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
20.00 µM |
CNE-2 |
Homo sapiens |
|
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT and STAT3 signaling pathways |
Western Blot |
10.00 mg/kg |
CNE-2 (xenograft) |
Mus musculus |
BALB/c nude |
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT and STAT3 signaling pathways |
Western Blot |
20.00 mg/kg |
CNE-2 (xenograft) |
Mus musculus |
BALB/c nude |
p-STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
1.25 µM |
CNE-2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
2.50 µM |
CNE-2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
5.00 µM |
CNE-2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
10.00 µM |
CNE-2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT pathway members |
Western Blot |
20.00 µM |
CNE-2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT and STAT3 signaling pathways |
Western Blot |
10.00 mg/kg |
CNE-2 (xenograft) |
Mus musculus |
BALB/c nude |
STAT3 |
|
Brevilin A |
Influence on PI3K/AKT and STAT3 signaling pathways |
Western Blot |
20.00 mg/kg |
CNE-2 (xenograft) |
Mus musculus |
BALB/c nude |
STAT3 |
|
Brevilin A |
Influence on STAT3 signalling |
Western Blot |
12.50 µM |
A549R |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on STAT3 signalling |
Western Blot |
25.00 µM |
A549R |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
5.00 µM |
DU145 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
10.00 µM |
DU145 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
15.00 µM |
DU145 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
5.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
10.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on constitutive STAT3 activation |
Western Blot |
15.00 µM |
MDA-MB-468 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein upon cytokine treatment |
Western Blot |
10.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein upon cytokine treatment |
Western Blot |
10.00 µM |
Hela |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein upon cytokine treatment |
Western Blot |
10.00 µM |
HepG2 |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on JAK2-JH1 overexpressed protein |
Western Blot |
10.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on JAK2-JH1 overexpressed protein |
Western Blot |
15.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein overexpression |
Western Blot |
15.00 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein overexpression |
Western Blot |
15.00 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein overexpression |
Western Blot |
15.00 µM |
HEK293T (JAK3-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on protein overexpression |
Western Blot |
15.00 µM |
HEK293T (Tyk2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain |
Western Blot |
10.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain |
Western Blot |
20.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain |
Western Blot |
40.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain |
Western Blot |
80.00 µM |
HEK293T |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
5.00 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
7.50 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
10.00 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
12.50 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
15.00 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
17.50 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
20.00 µM |
HEK293T (JAK1-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
5.00 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
7.50 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
10.00 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
12.50 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
15.00 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
17.50 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
20.00 µM |
HEK293T (JAK2-JH1) |
Homo sapiens |
|
STAT3 |
|
Brevilin A |
Measurement of IC50 value JAKs-JH1 truncated kinases |
Western Blot |
5.00 µM |
HEK293T (JAK3-JH1) |
Homo sapiens |
|
STAT3 |
|