| AZD1480 |
Influence on protein activity |
Western Blot |
0.50 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
2.50 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
5.00 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
0.50 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
2.50 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
5.00 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
0.50 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
2.50 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
5.00 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
0.50 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
2.50 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
5.00 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
0.50 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
1.00 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
2.50 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
5.00 µM |
KCNR |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
0.50 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
1.00 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
2.50 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
5.00 µM |
SY5Y |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
0.50 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
1.00 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
2.50 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
5.00 µM |
Rh18 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
0.50 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
1.00 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
2.50 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of IL-6 |
Western Blot |
5.00 µM |
TC32 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
KCNR (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
SY5Y (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
Rh18 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
TC32 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on late protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
KCNR (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on late protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
SY5Y (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on late protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
Rh18 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on late protein activity in tumor tissue |
Western Blot |
30.00 mg/kg |
TC32 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
U251-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity |
Western Blot |
1.00 µM |
U87-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Cell Apoptosis Analysis |
Western Blot |
1.00 µM |
U251-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Cell Apoptosis Analysis |
Western Blot |
10.00 µM |
U251-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
0.10 µM |
U87-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
0.50 µM |
U87-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
1.00 µM |
U87-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
10.00 µM |
U87-MG |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
0.10 µM |
4C8 |
Homo sapiens |
|
|
|
| AZD1480 |
Influence on protein activity in presence of OSM |
Western Blot |
0.50 µM |
4C8 |
Homo sapiens |
|
|
|
