S3I-M2001 |
Influence on tumor growth |
Tumor volume |
5.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
S3I-M2001 |
Influence on tumor growth |
Tumor volume |
10.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
S3I-M2001 |
Influence on tumor growth |
Tumor volume |
20.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
|
|
S3I-M2001 |
Influence on DNA binding in tumor |
EMSA |
5.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
STAT3:STAT3 |
|
S3I-M2001 |
Influence on protein activity in tumor tissue |
Western Blot |
5.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
STAT3 |
|
S3I-M2001 |
Influence on protein activity in tumor tissue |
Western Blot |
5.00 mg/kg |
MDA-MB-231 (xenograft) |
Mus musculus |
athymic nude mice |
p-STAT3(Y705) |
|