Investigated event: Influence on protein activity

Name Value
Compound SD-91
Investigated event Influence on protein activity
Experiment type Western Blot
Concentration 6.25 µM
Cell line SUP-M2
Organism Homo sapiens
Animal model
STAT protein STAT3
Other
Reference
SD-91 as A Potent and Selective STAT3 Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression. ACS medicinal chemistry letters Haibin Zhou, Longchuan Bai, Renqi Xu, Donna McEachern, Krishnapriya Chinnaswamy, Ruiting Li, Bo Wen, Mi Wang, Chao-Yie Yang, Jennifer L Meagher, Duxin Sun, Jeanne A Stuckey, Shaomeng Wang, 12, 6, 2021-06-10, 2021-05-10, 10.1021/acsmedchemlett.1c00155 DOI: 10.1021/acsmedchemlett.1c00155 PUBMED: 34141084 PMCID: PMC8201759