CJ-1383

Name	Value
Weight	0.000 g/mol
Zinc ID	N/A
Smiles	N/A
Molecular formula	N/A
Mode of inhibition	Direct STAT SH2; Peptidomimetic
CAS	GLXC-21813

Clinical Trials

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References

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Publication	DOI	Pubmed	PMCID
Structure-Based Design of Conformationally Constrained, Cell-Permeable STAT3 Inhibitors. ACS medicinal chemistry letters Jianyong Chen, Longchuan Bai, Denzil Bernard, Zaneta Nikolovska-Coleska, Cindy Gomez, Jian Zhang, Han Yi, Shaomeng Wang, 1, 2, 2010-05-13, None, 10.1021/ml100010j	10.1021/ml100010j	20596242	PMC2892918

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Filter data

Compound	CJ-1383
Experiment types	Flow cytometry , Fluorescence polarization assay, Western Blot
Concentrations	1.25, 10.00, 2.50, 20.00, 5.00, N/A
Cell lines	MDA-MB-468
Organisms	Homo sapiens
Animal models
STAT proteins	STAT3, p-STAT3
Other	Bcl-xL, Cas-3, Cleaved Cas-3, Cleaved-PARP, Cyclin D1, GAPDH, PARP

Experiments

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Compound	Experiment type	Investigated event	Concentration	Cell line	Organism	Animal model	Stat protein	Details
CJ-1383	Fluorescence polarization assay	Protein binding activity	N/A µM		Homo sapiens
CJ-1383	Flow cytometry	Influence on cell apoptosis	20.00 µM	MDA-MB-468	Homo sapiens
CJ-1383	Flow cytometry	Influence on cell apoptosis	10.00 µM	MDA-MB-468	Homo sapiens
CJ-1383	Flow cytometry	Influence on cell apoptosis	5.00 µM	MDA-MB-468	Homo sapiens
CJ-1383	Flow cytometry	Influence on cell apoptosis	2.50 µM	MDA-MB-468	Homo sapiens
CJ-1383	Western Blot	Influence on protein activity	20.00 µM	MDA-MB-468	Homo sapiens		STAT3
CJ-1383	Western Blot	Influence on protein activity	10.00 µM	MDA-MB-468	Homo sapiens		STAT3
CJ-1383	Western Blot	Influence on protein activity	5.00 µM	MDA-MB-468	Homo sapiens		STAT3
CJ-1383	Western Blot	Influence on protein activity	2.50 µM	MDA-MB-468	Homo sapiens		STAT3
CJ-1383	Western Blot	Influence on protein activity	1.25 µM	MDA-MB-468	Homo sapiens		STAT3

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