Baricitinib (INCB028050)

Name Value
Weight 371.426 g/mol
Zinc ID ZINC73069247
Smiles CCS(=O)(=O)N1CC(CC#N)(n2cc(-c3ncnc4[nH]ccc34)cn2)C1
Molecular formula C16H17N7O2S
Mode of inhibition N/A
CAS 1187594-09-7

Clinical Trials

Study title Status Conditions Link
Baricitinib in the Treatment of Adults With Pyoderma Gangrenosum (PG) Recruiting Pyoderma Gangrenosum|Skin Diseases|Wound Heal|Pyoderma|Skin Ulcer NCT04901325
A Study of Baricitinib (LY3009104) in Children With COVID-19 (COV-BARRIER-PEDS) Not yet recruiting Covid19|Corona Virus Infection NCT05074420
Baricitinib Therapy in COVID-19 Completed COVID|Pneumonia NCT04358614
Baricitinib for the Prophylaxis of Graft-Versus-Host Disease After Peripheral Blood Hematopoietic Cell Transplantation Recruiting Graft-versus-host-disease|Graft Vs Host Disease NCT04131738
Baricitinib for coRona Virus pnEumonia (COVID-19): a THerapeutic Trial Not yet recruiting Corona Virus Infection NCT04399798
A Study of Baricitinib (LY3009104) in Adult and Pediatric Japanese Participants With NNS/CANDLE, SAVI, and AGS Active, not recruiting Nakajo-Nishimura Syndrome|Chronic Atypical Neutrophilic Dermatosis With Lipodystrophy and Elevated Temperature Syndrome|STING-Associated Vasculopathy With Onset in Infancy|Aicardi Goutieres Syndrome NCT04517253
A Study of Baricitinib in Healthy Participants Completed Healthy NCT03212638
Safety and Efficacy of Baricitinib for COVID-19 Withdrawn COVID-19 NCT04340232
A Study to Measure Baricitinib (LY3009104) Absorption in Healthy Participants Completed Healthy Volunteers NCT02340104
A Study of Baricitinib in Participants From 1 Year to Less Than 18 Years Old With Juvenile Idiopathic Arthritis Recruiting Juvenile Idiopathic Arthritis NCT03773965
A Study of Baricitinib (LY3009104) in Participants With Moderate to Severe Atopic Dermatitis Active, not recruiting Atopic Dermatitis NCT03559270
A Study of Baricitinib (LY3009104) in Adult Participants With Moderate to Severe Atopic Dermatitis Completed Atopic Dermatitis NCT03435081
A Study of Baricitinib in Participants With Systemic Lupus Erythematosus (SLE) Recruiting Systemic Lupus Erythematosus NCT03843125
Study of Baricitinib (LY3009104) in Patients With Moderate to Severe Atopic Dermatitis Completed Atopic Dermatitis NCT03334422
Baricitinib in Patients With Relapsing or naĂŻve Dermatomyositis Not yet recruiting Dermatomyositis NCT04972760
JAK Inhibitor Treatment in AGS Active, not recruiting Aicardi Goutieres Syndrome NCT03921554
A Pharmacokinetic Study of Baricitinib in Participants With Liver Disease Completed Liver Diseases|Hepatic Insufficiency NCT01870388
Baricitinib in Relapsing Giant Cell Arteritis Completed Arteritis, Giant Cell NCT03026504
A Study of Baricitinib (LY3009104) in Participants From 1 Year to Less Than 18 Years Old With sJIA Recruiting Systemic Juvenile Idiopathic Arthritis NCT04088396
Efficacy and Safety of Baricitinib in Sjogren's Syndrome Not yet recruiting Sjogren's Syndrome NCT05016297
Effect of Baricitinib Treatment on Peripheral Bone in RA Active, not recruiting Rheumatoid Arthritis|Bone Density|Finger Joints NCT03701789
A Study of Baricitinib and Ciclosporin in Healthy Participants Completed Healthy Volunteers NCT01968057
A Prospective Pilot Study to Explore Efficacy and Safety of Baricitinib in Active Primary Sjogren's Syndrome Patients Completed Sjogren's Syndrome NCT04916756
A Study of Baricitinib (LY3009104) in Participants With COVID-19 Completed COVID-19 NCT04421027
A Study of Baricitinib (LY3009104) in Healthy Chinese Participants Completed Healthy NCT02758613
A Study of Baricitinib and Omeprazole in Healthy Participants Completed Healthy Volunteers NCT01925144
Tocilizumab Versus Baricitinib in Patients With Severe COVID-19 Recruiting COVID-19 NCT05082714
A Study of Baricitinib and Rifampicin in Healthy Participants Completed Healthy Volunteers NCT01910311
Efficacy and Safety of Baricitinib in Patients With Moderate and Severe COVID-19 Not yet recruiting Covid19 NCT05056558
Baricitinib in Symptomatic Patients Infected by COVID-19: an Open-label, Pilot Study. Not yet recruiting Pharmacological Action NCT04320277
A Study of Baricitinib in Healthy Japanese Participants Completed Healthy Participants NCT02263911
A Study of Baricitinib (LY3009104) in Children and Adolescents With Atopic Dermatitis Recruiting Atopic Dermatitis NCT03952559
A Study of Baricitinib in Participants From 2 Years to Less Than 18 Years Old With Juvenile Idiopathic Arthritis Active, not recruiting Juvenile Idiopathic Arthritis NCT03773978
A Study of Baricitinib (LY3009104) in Patients With Moderate to Severe Atopic Dermatitis Completed Atopic Dermatitis NCT03334396
A Study of Baricitinib in Participants With Systemic Lupus Erythematosus Completed Systemic Lupus Erythematosus NCT03616964
A Study of Baricitinib (LY3009104) in Participants With Systemic Lupus Erythematosus Completed Systemic Lupus Erythematosus NCT03616912
A Long-term Study of Baricitinib (LY3009104) With Topical Corticosteroids in Adults With Moderate to Severe Atopic Dermatitis That Are Not Controlled With Cyclosporine or for Those Who Cannot Take Oral Cyclosporine Because it is Not Medically Advisable Active, not recruiting Atopic Dermatitis NCT03428100
A Study of Baricitinib (LY3009104) in Participants From 2 Years to Less Than 18 Years Old With Active JIA-Associated Uveitis or Chronic Anterior Antinuclear Antibody-Positive Uveitis Recruiting Uveitis NCT04088409
A Study of Baricitinib (LY3009104) in Adults With Severe or Very Severe Alopecia Areata Active, not recruiting Alopecia Areata NCT03899259
Baricitinib in New-onset Type 1 Diabetes Recruiting Type 1 Diabetes NCT04774224
Study of Baricitinib, a JAK1/2 Inhibitor, in Chronic Graft-Versus-Host Disease After Allogeneic Hematopoietic Stem Cell Transplantation Active, not recruiting Chronic Graft vs Host Disease|Chronic Graft-Versus-Host Disease NCT02759731
A Study of Baricitinib in Participants With Rheumatoid Arthritis Recruiting Rheumatoid Arthritis NCT04086745
A Study of Baricitinib (LY3009104) in Participants With Systemic Lupus Erythematosus (SLE) Completed Systemic Lupus Erythematosus NCT02708095
Exploiting Leading Edge 7T MRI Brain Imaging to Decipher Olumiant's Mode of Analgesic Action in Rheumatoid Arthritis Recruiting Rheumatoid Arthritis NCT05112120
A Study of Baricitinib (LY3009104) in Participants With Severe or Very Severe Alopecia Areata Active, not recruiting Alopecia Areata NCT03570749
A Study of Baricitinib (LY3009104) in Participants With Rheumatoid Arthritis Active, not recruiting Rheumatoid Arthritis NCT03915964
A Study of Baricitinib and Probenecid in Healthy Participants Completed Healthy Volunteers NCT01937026
A Study of Baricitinib and Birth Control Pills in Healthy Females Completed Healthy Volunteers NCT01896726
A Drug Drug Interaction (DDI) Study of Baricitinib (LY3009104) and Digoxin in Healthy Participants Completed Healthy Volunteers NCT01859078
A Study of Baricitinib When Administered With Ketoconazole or Fluconazole in Healthy Participants Completed Healthy Volunteers NCT01924299
Combination of Baricitinib and Adalimumab in Rheumatoid Arthritis Recruiting Rheumatoid Arthritis NCT04870203
A Phase 2b Study of Baricitinib in Participants With Moderate to Severe Psoriasis Completed Psoriasis|Skin Diseases|Skin Diseases, Papulosquamous NCT01490632
Baricitinib Compared to Standard Therapy in Patients With COVID-19 Not yet recruiting Covid-19|SARS-CoV 2|SARS Pneumonia NCT04393051
A Study of Baricitinib (LY3009104) in Participants With Rheumatoid Arthritis (RA) Completed Rheumatoid Arthritis NCT02265705
A Study of Baricitinib (LY3009104) in Participants With Primary Biliary Cholangitis Who do Not Respond or Cannot Take UDCA Terminated Primary Biliary Cholangitis NCT03742973
Efficacy of Baricitinib In Treatment of Delayed-Type Hypersensitivity Versus Irritant Skin Reactions in Healthy Adult Male Subjects Recruiting Allergic Contact Dermatitis NCT03945760
A Study of Baricitinib (LY3009104) in Combination With Topical Corticosteroids in Adults With Moderate to Severe Atopic Dermatitis Completed Atopic Dermatitis NCT03733301
Efficacy of Ramdicivir and Baricitinib for the Treatment of Severe COVID 19 Patients Recruiting Covid19|Covid-19 ARDS NCT04693026
Baricitinib in Hospitalized Covid-19 Patients With Diabetes Mellitus Recruiting COVID-19 Pneumonia NCT04970719
Evaluation of Effect and Tolerance of the Association of Baricitinib and Phototherapy Versus Phototherapy in Adults With Progressive Vitiligo Not yet recruiting Vitiligo NCT04822584
A Study of Baricitinib and Simvastatin in Healthy Participants Completed Healthy Volunteers NCT01960140
Baricitinib, Placebo and Antiviral Therapy for the Treatment of Patients With Moderate and Severe COVID-19 Terminated Symptomatic COVID-19 Infection Laboratory-Confirmed NCT04373044
A Study of Long-term Baricitinib (LY3009104) Therapy in Atopic Dermatitis Active, not recruiting Atopic Dermatitis NCT03334435
A Study of Baricitinib (LY3009104) in Participants With Moderate-to-Severe Atopic Dermatitis Completed Atopic Dermatitis NCT02576938
Disposition of 14C-LY3009104 Following Oral Administration in Healthy Human Subjects Completed Healthy Volunteers NCT01299285
A Moderate to Severe Rheumatoid Arthritis Study Completed Rheumatoid Arthritis NCT01721044
Bioequivalence Study of Baricitinib From Barcimiant 4 mg Film Coated Tablets (Horus Pharma, Egypt) and Olumiant 4 mg Film Coated Tablets (Eli Lilly Nederland B.V., The Netherlands) Completed Healthy NCT05006768
A Study to Test Safety and Efficacy of Baricitinib in Participants With Diabetic Kidney Disease Completed Diabetic Kidney Disease NCT01683409
Factorial Randomized Trial of Rendesivir and Baricitinib Plus Dexamethasone for COVID-19 (the AMMURAVID Trial) Not yet recruiting Covid19 NCT04832880
An Extension Study in Participants With Moderate to Severe Rheumatoid Arthritis Completed Rheumatoid Arthritis NCT01885078
Examination of Efficacy and Safety of Baricitinib in RA Patients Recruiting Rheumatoid Arthritis NCT03755466
BAriCitinib Healing Effect in earLy pOlymyalgia Rheumatica Recruiting Polymyalgia Rheumatic (PMR) NCT04027101
A Study of LY3009104(Baricitinib) for Healthy Subjects Completed Healthy Volunteer NCT01247350
JAK 1/2 Inhibitor, Baricitinib, in the Treatment of Adult IIM Recruiting Idiopathic Inflammatory Myopathies NCT04208464
A Study of LY3009104 in Healthy Participants Completed Healthy Participants NCT01536951
A Study in Participants With Moderate to Severe Rheumatoid Arthritis Completed Rheumatoid Arthritis NCT01711359
Oral Baricitinib (LY3009104)Treatment in Japanese Participants With Active Rheumatoid Arthritis on Background Methotrexate Therapy Completed Arthritis, Rheumatoid NCT01469013
A Study in Moderate to Severe Rheumatoid Arthritis Participants Completed Rheumatoid Arthritis NCT01721057
A Study in Moderate to Severe Rheumatoid Arthritis Completed Rheumatoid Arthritis NCT01710358
INCB028050 Compared to Background Therapy in Patients With Active Rheumatoid Arthritis (RA) With Inadequate Response to Disease Modifying Anti-Rheumatic Drugs Completed Rheumatoid Arthritis NCT00902486
Clinical Trial to Evaluate Efficacy of 3 Types of Treatment in Patients With Pneumonia by COVID-19 Active, not recruiting COVID-19 Pneumonia NCT04346147
Clinical-epidemiological Characterization of COVID-19 Disease in Hospitalized Older Adults Completed COVID-19 NCT04362943
A Relative Bioavailability and Food Effect Study of New Formulations Completed Chronic Inflammatory Disorder|Arthritis, Rheumatoid NCT01398475
mulTi-Arm Therapeutic Study in Pre-ICu Patients Admitted With Covid-19 - Repurposed Drugs (TACTIC-R) Recruiting COVID19 NCT04390464
EU SolidAct: An Adaptive Pandemic and Emerging Infection Platform Trial Recruiting COVID-19|Emerging Infectious Disease NCT04891133
Adaptive COVID-19 Treatment Trial 2 (ACTT-2) Completed COVID-19 NCT04401579
A Study in Participants With Rheumatoid Arthritis on Background Methotrexate Therapy Completed Arthritis, Rheumatoid NCT01185353
Adaptive COVID-19 Treatment Trial 4 (ACTT-4) Completed COVID-19 NCT04640168
Treatment of Moderate to Severe Coronavirus Disease (COVID-19) in Hospitalized Patients Recruiting COVID-19 NCT04321993
Compassionate Use Protocol for the Treatment of Autoinflammatory Syndromes No longer available Chronic Atypical Neutrophilic Dermatosis With Lipodystrophy and Elevated Temperature (CANDLE)|Juvenile Dermatomyositis (JDM)|Stimulator of Interferon Genes (STING)-Associated Vasculopathy With Onset During Infancy (SAVI)|Aicardi-Goutières Syndrome (AGS) NCT01724580
Comparative Effectiveness of Targeted Therapy in RA Patients Recruiting Rheumatoid Arthritis NCT04449224
Clinical Trial to Evaluate the Efficacy of Different Treatments in Patients With COVID-19 Recruiting SARS-CoV-2 Infection NCT04890626
Randomised Evaluation of COVID-19 Therapy Recruiting Severe Acute Respiratory Syndrome NCT04381936
Splenic Stimulation for RA Recruiting Rheumatoid Arthritis NCT05003310
Microbiome in Atopic Dermatitis Under Systemic Therapy Recruiting Atopic Dermatitis NCT05099315
Screening for Flare After b/tsDMARD Discontinuation in Rheumatoid Arthritis Not yet recruiting Rheumatoid Arthritis NCT05119452
Effects of Antirheumatic Treatment on Levels of Survivin in Rheumatoid Arthritis Patients Recruiting Rheumatoid Arthritis NCT03440892
Effect of Treatments in Patients Hospitalized for Severe COVID-19 Pneumonia: a Multicenter Cohort Study Recruiting Covid-19|ARDS|Pneumonia NCT04365764
Factors Associated With Clinical Outcomes in Patients Hospitalized for Covid-19 in GHT-93 Est Recruiting COVID|SARS-CoV 2 NCT04366206
Effect of Antiinflammatory Treatment Versus Hand Training on Neuropsychiatric Comorbidity in RA-patients Recruiting Rheumatoid Arthritis|Pain|Fatigue|Cognitive Decline|Depression|Brain Diseases|Hand Rheumatism NCT04378621
Evaluation of Pain Sensitization in Rheumatoid Arthritis: Analysis on a Cohort of Tofacitinib Treated Patients Recruiting Rheumatoid Arthritis NCT03815578
Microbiota Analysis to Predict Outcomes of Rheumatoid Arthritis Patients Treated With JAK-inhibitor Recruiting Rheumatoid Arthritis NCT04530305
Molecular Signatures in Inflammatory Skin Disease Recruiting Atopic Dermatitis|Psoriasis NCT03358693
Results in Real Clinical Practice of Treatment of Moderate-severe Atopic Dermatitis Recruiting Dermatitis, Atopic NCT05078294
JAKPOT (JAK Inhibitors and Predictors of Outcome in rheumaToid Arthritis) Recruiting Rheumatoid Arthritis NCT04084223
Treatment of Rheumatoid Arthritis With DMARDs: Predictors of Response Recruiting Rheumatoid Arthritis NCT03414502
Immunopathology of Polymyalgia Rheumatica on Shoulder Bursae's Biopsies Not yet recruiting Polymyalgia Rheumatica NCT04727879

References

Publication DOI Pubmed PMCID

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Compound Baricitinib (INCB028050)
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Experiments

Compound Experiment type Investigated event Concentration Cell line Organism Animal model Stat protein Details